Synthesis and cytotoxicity testing of new amido-substituted triazolopyrrolo[2,1-c][1,4]benzodiazepine (PBDT) derivatives.

نویسندگان

  • Kumaraswamy Sorra
  • Chi-Fen Chang
  • Srinivas Pusuluri
  • Khagga Mukkanti
  • Min-Chiau Laiu
  • Bo-Ying Bao
  • Chia-Hao Su
  • Ta-Hsien Chuang
چکیده

A series of amido-substituted triazolopyrrolo[2,1-c][1,4]benzodiazepine (PBDT) derivatives was synthesized from isatoic anhydride, and their cytotoxicity against the MRC-5 and Mahlavu cell lines was evaluated. The results suggest that compound PBDT-7i with the meta-trifluoromethylbenzoyl substituent can selectively inhibit the growth of Mahlavu cells and has low toxicity towards MRC-5 cells.

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عنوان ژورنال:
  • Molecules

دوره 17 8  شماره 

صفحات  -

تاریخ انتشار 2012